Receptor Ligands
Agonists :
5-FNE •
6-FNE •
Amidephrine •
Anisodamine •
Anisodine •
Cirazoline •
Dipivefrine •
Dopamine •
Ephedrine •
Epinephrine (Adrenaline) •
Etilefrine •
Ethylnorepinephrine •
Indanidine •
Levonordefrin •
Metaraminol •
Methoxamine •
Methyldopa •
Midodrine •
Naphazoline •
Norepinephrine (Noradrenaline) •
Octopamine •
Oxymetazoline •
Phenylephrine •
Phenylpropanolamine •
Pseudoephedrine •
Synephrine •
Tetrahydrozoline Antagonists :
Abanoquil •
Adimolol •
Ajmalicine •
Alfuzosin •
Amosulalol •
Arotinolol •
Atiprosin •
Benoxathian •
Buflomedil •
Bunazosin •
Carvedilol •
CI-926 •
Corynanthine •
Dapiprazole •
DL-017 •
Domesticine •
Doxazosin •
Eugenodilol •
Fenspiride •
GYKI-12,743 •
GYKI-16,084 •
Indoramin •
Ketanserin •
L-765,314 •
Labetalol •
Mephendioxan •
Metazosin •
Monatepil •
Moxisylyte (Thymoxamine) •
Naftopidil •
Nantenine •
Neldazosin •
Nicergoline •
Niguldipine •
Pelanserin •
Phendioxan •
Phenoxybenzamine •
Phentolamine •
Piperoxan •
Prazosin •
Quinazosin •
Ritanserin •
RS-97,078 •
SGB-1,534 •
Silodosin •
SL-89.0591 •
Spiperone •
Talipexole •
Tamsulosin •
Terazosin •
Tibalosin •
Tiodazosin •
Tipentosin •
Tolazoline •
Trimazosin •
Upidosin •
Urapidil •
Zolertine * Note that many TCAs , TeCAs , antipsychotics , ergolines , and some piperazines like buspirone , trazodone , nefazodone , etoperidone , and mepiprazole all antagonize α1 -adrenergic receptors as well, which contributes to their side effects such as orthostatic hypotension .
Reuptake Inhibitors
Releasing Agents مستقبلات الإنزيمات
أخرى
Receptor Ligands
Benzazepines :
6-Br-APB •
Fenoldopam •
SKF-38,393 •
SKF-77,434 •
SKF-81,297 •
SKF-82,958 •
SKF-83,959 ;
Ergot-derivatives :
Bromocriptine •
Cabergoline •
Dihydroergocryptine •
Lisuride •
LSD •
Pergolide ;
Dihydrexidine-derivatives :
A-86,929 •
Dihydrexidine •
Dinapsoline •
Dinoxyline •
Doxanthrine ;
Morphine-derivatives :
Apomorphine •
Propylnorapomorphine ;
Piperazines :
ABT-724 •
Aripiprazole •
Piribedil •
WAY-100,635 ;
Others :
7-OH-DPAT •
A-68,930 •
A-77,636 •
A-412,997 •
Amantadine •
Aplindore •
CY-208,243 •
Memantine •
Pramipexole •
Pukateine •
Quinpirole •
RDS-127 •
Rimantadine •
Ropinirole •
Rotigotine
Reuptake Inhibitors
Releasing Agents Oxazolines :
4-Methylaminorex (4-MAR, 4-MAX) •
Aminorex •
Clominorex •
Cyclazodone •
Fenozolone •
Fluminorex •
Pemoline •
Thozalinone ;
Phenethylamines (also
Amphetamines ,
Cathinones ,
Phentermines , etc):
2-Hydroxyphenethylamine (2-OH-PEA) •
4-Methylamphetamine (4-MA) •
4-Methylmethamphetamine (4-MMA) •
α-Ethylphenethylamine (α-Et-PEA) •
Alfetamine •
Amphetamine (
Dextroamphetamine ,
Levoamphetamine ) •
Amphetaminil •
Amfepentorex •
β-Methylphenethylamine (β-Me-PEA) •
Benzodioxolylbutanamine (BDB) •
Benzodioxolylhydroxybutanamine (BOH) •
Benzphetamine •
Brephedrone •
Butylone •
Cathine •
Cathinone •
Clephedrone •
Clobenzorex •
Clortermine •
Diethylcathinone (Diethylpropion, Amfepramone) •
Dibutylone •
Dimethoxyamphetamine (DMA) •
Dimethoxymethamphetamine (DMMA) •
Dimethylamphetamine •
Dimethylcathinone (Dimethylpropion, Metamfepramone) •
Ethcathinone (Ethylpropion) •
Ethylamphetamine •
Ethylbenzodioxolylbutanamine (EBDB) •
Ethylone •
Fenethylline •
Fenproporex •
Flephedrone •
Fludorex •
Furfenorex •
Hordenine •
Indanorex •
Indanylamphetamine (IAP) •
Iodephedrone •
Lisdexamfetamine •
Lophophine (Homomyristicylamine) •
Mefenorex •
Mephedrone •
Methamphetamine (Desoxyephedrine, Methedrine;
Dextromethamphetamine ,
Levomethamphetamine ) •
Methcathinone (Methylpropion) •
Methedrone •
Methoxymethylenedioxyamphetamine (MMDA) •
Methoxymethylenedioxymethamphetamine (MMDMA) •
Methylbenzodioxolylbutanamine (MBDB) •
Methylenedioxyamphetamine (MDA; Tenamfetamine) •
Methylenedioxyethylamphetamine (MDEA) •
Methylenedioxyhydroxyamphetamine (MDOH) •
Methylenedioxymethamphetamine (MDMA) •
Methylenedioxymethylphenethylamine (MDMPEA; Homarylamine) •
Methylenedioxyphenethylamine (MDPEA; Homopiperonylamine) •
Methylone •
Naphthylamphetamine (NAP) •
Ortetamine •
Oxaflozane •
Parabromoamphetamine (PBA) •
Parachloroamphetamine (PCA) •
Parafluoroamphetamine (PFA) •
Parafluoromethamphetamine (PFMA) •
Parahydroxyamphetamine (PHA) •
Paraiodoamphetamine (PIA) •
Paramethoxyamphetamine (PMA) •
Paramethoxyethylamphetamine (PMEA) •
Paramethoxymethamphetamine (PMMA) •
Paredrine (Norpholedrine, Oxamphetamine) •
Phendimetrazine •
Phenethylamine (PEA) •
Phenmetrazine •
Pholedrine •
Phenpromethamine •
Propylamphetamine •
Tiflorex (Flutiorex) •
Tyramine (TRA) •
Xylopropamine •
Zylofuramine ;
Piperazines :
2,5-Dimethoxy-4-bromobenzylpiperazine (2C-B-BZP) •
Benzylpiperazine (BZP) •
Methoxyphenylpiperazine (MeOPP; Paraperazine) •
Methylbenzylpiperazine (MBZP) •
Methylenedioxybenzylpiperazine (MDBZP; Piperonylpiperazine);
Others :
2-Aminoindane (2-AI) •
2-Aminotetralin (2-AT) •
4-Benzylpiperidine (4-BP) •
Clofenciclan •
Cyclopentamine •
Cypenamine •
Cyprodenate •
Feprosidnine •
Gilutensin •
Heptaminol •
Hexacyclonate •
Isometheptene •
Methylhexanamine •
Octodrine •
Phthalimidopropiophenone •
Propylhexedrine (PHX) •
Tuaminoheptane (Tuamine)
Enzyme Inhibitors
Others
Receptor Ligands
Agonists :
Lysergamides :
Dihydroergotamine •
Methysergide ;
Triptans :
Almotriptan •
Eletriptan •
Frovatriptan •
Naratriptan •
Rizatriptan •
Sumatriptan •
Zolmitriptan ;
Tryptamines :
5-CT •
5-MT ;
Others :
CP-135,807 •
CP-286,601 •
GR-46611 •
L-694,247 •
L-772,405 •
PNU-109,291 •
PNU-142,633 Antagonists :
Lysergamides :
Metergoline •
Methiothepin ;
Tryptamines :
Rauwolscine •
Yohimbine ;
Others :
BRL-15572 •
GR-127,935 •
Ketanserin •
LY-310,762 •
LY-367,642 •
LY-456,219 •
LY-456,220 •
Ritanserin •
Ziprasidone
Agonists :
Phenethylamines :
2C-B •
2C-E •
2C-I •
2C-T-2 •
2C-T-7 •
2C-T-21 •
DOB •
DOC •
DOI •
DOM •
MDA •
MDMA •
Mescaline •
Myristicin ;
Piperazines :
Aripiprazole •
mCPP •
TFMPP ;
Tryptamines :
5-CT •
5-MeO-α-ET •
5-MeO-α-MT •
5-MeO-DET •
5-MeO-DiPT •
5-MeO-DMT •
5-MeO-DPT •
5-MT •
α-ET •
α-Methyl-5-HT •
α-MT •
Bufotenin •
DET •
DiPT •
DMT •
DPT •
Psilocin •
Psilocybin ;
Others :
A-372,159 •
AL-38022A •
CP-809,101 •
Lorcaserin •
MK-212 •
PNU-22394 •
Ro60-0175 •
Vabicaserin •
WAY-629 •
WAY-161,503 •
YM-348 Antagonists :
Atypical Antipsychotics :
Clozapine •
Iloperidone •
Melperone •
Olanzapine •
Paliperidone •
Pimozide •
Quetiapine •
Risperidone •
Sertindole •
Ziprasidone •
Zotepine ;
Typical Antipsychotics :
Loxapine •
Pipamperone ;
Antidepressants :
Agomelatine •
Amitriptyline •
Amoxapine •
Etoperidone •
Fluoxetine •
Mianserin •
Mirtazapine •
Nefazodone •
Trazodone ;
Others :
Cinanserin •
Deramciclane •
Dimebolin •
Dotarizine •
Eltoprazine •
FR-260,010 •
Ketanserin •
Pizotifen •
Ritanserin •
RS-102,221 •
SB-200,646 •
SB-206,553 •
SB-221,284 •
SB-228,357 •
SB-242,084 •
SB-243,213 •
SDZ SER-082 •
Xylamidine
5-HT5B *
Agonists :
Lysergamides :
Ergotamine •
LSD Antagonists :
Methiothepin * Note that the 5-HT5B receptor is not functional in humans.
Reuptake Inhibitors
Releasing Agents Enzyme Inhibitors
Others